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James Papatzimas
James Papatzimas
Novartis Institute for BioMedical Research
Verified email at novartis.com
Title
Cited by
Cited by
Year
From inhibition to degradation: targeting the antiapoptotic protein myeloid cell leukemia 1 (MCL1)
JW Papatzimas, E Gorobets, R Maity, MI Muniyat, JL MacCallum, P Neri, ...
Journal of Medicinal Chemistry 62 (11), 5522-5540, 2019
932019
Rational chemical design of molecular glue degraders
ES Toriki, JW Papatzimas, K Nishikawa, D Dovala, AO Frank, MJ Hesse, ...
ACS central science 9 (5), 915-926, 2023
432023
Thiaporphyrin-mediated photocatalysis using red light
JG Lee, JW Papatzimas, AD Bromby, E Gorobets, DJ Derksen
RSC advances 6 (64), 59269-59272, 2016
272016
A facile synthesis of ligands for the von Hippel–Lindau E3 ligase
C Steinebach, SA Voell, LP Vu, A Bricelj, I Sosič, G Schnakenburg, ...
Synthesis 52 (17), 2521-2527, 2020
232020
ADAM protease inhibition overcomes resistance of breast cancer stem-like cells to γδ T cell immunotherapy
I Dutta, D Dieters-Castator, JW Papatzimas, A Medina, J Schueler, ...
Cancer letters 496, 156-168, 2021
142021
A general strategy for the preparation of thalidomide-conjugate linkers
JW Papatzimas, E Gorobets, DK Brownsey, R Maity, NJ Bahlis, ...
Synlett 28 (20), 2881-2885, 2017
132017
Identification of ligand linkage vectors for the development of p300/CBP degraders
DK Brownsey, BC Rowley, E Gorobets, K Mihara, R Maity, JW Papatzimas, ...
RSC Medicinal Chemistry 13 (6), 726-730, 2022
42022
A vinylogous Norrish reaction as a strategy for light-mediated ring expansion
E Gorobets, JW Papatzimas, J Dourado, G Yousefalizadeh, JG Lee, ...
Chemical Communications 58 (17), 2910-2913, 2022
32022
Sulfamoyl benzene derivatives and uses thereof
T Trang, DJ Derksen, K Navis, E Gorobets, J Papatzimas
US Patent App. 18/024,443, 2024
2024
DCAF16-Based Covalent Handle for the Rational Design of Monovalent Degraders
M Lim, TD Cong, LM Orr, ES Toriki, AC Kile, JW Papatzimas, E Lee, Y Lin, ...
ACS Central Science, 2024
2024
Correction to “Rational Chemical Design of Molecular Glue Degraders”
ES Toriki, JW Papatzimas, K Nishikawa, D Dovala, AO Frank, MJ Hesse, ...
ACS Central Science 9 (8), 1702-1702, 2023
2023
Correction to “Rational Chemical Design of Molecular Glue Degraders”
DK Nomura, ES Toriki, JW Papatzimas, K Nishikawa, D Dovala, AO Frank, ...
ACS Central Science 9 (8), , 1702, 2023
2023
Rational Chemical Design of Molecular Glue Degraders
J McKenna, D Dovala, A Frank, M Hesse, J Song, M Bruce-Smythe, ...
ACS Central Science, 2023
2023
Synthesis and Biological Evaluation of Heterobifunctional Small Molecules for Proteasome-Mediated Protein Degradation of Myeloid Cell Leukemia 1 (MCL1)
JW Papatzimas
Synthesis 2020, 09-14, 2020
2020
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