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| Amide-to-ester substitution as a strategy for optimizing PROTAC permeability and cellular activity VG Klein, AG Bond, C Craigon, RS Lokey, A Ciulli Journal of medicinal chemistry 64 (24), 18082-18101, 2021 | 77 | 2021 |
| Development of BromoTag: a “bump-and-hole”–PROTAC system to induce potent, rapid, and selective degradation of tagged target proteins AG Bond, C Craigon, KH Chan, A Testa, A Karapetsas, R Fasimoye, ... Journal of Medicinal Chemistry 64 (20), 15477-15502, 2021 | 47 | 2021 |
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| Targeting epigenetic modulators using PROTAC degraders: Current status and future perspective T Webb, C Craigon, A Ciulli Bioorganic & Medicinal Chemistry Letters 63, 128653, 2022 | 22 | 2022 |
| Targeted protein degradation via intramolecular bivalent glues O Hsia, M Hinterndorfer, AD Cowan, K Iso, T Ishida, R Sundaramoorthy, ... Nature, 1-8, 2024 | 10 | 2024 |
| An intramolecular bivalent degrader glues an intrinsic BRD4-DCAF16 interaction O Hsia bioRxiv, 2023 | 9 | 2023 |
| Development and application of BromoTag, a" bump-&-hole"-PROTAC degron system for rapid, potent, and selective degradation of tagged target proteins CG Craigon University of Dundee, 2022 | | 2022 |
