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Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity MKW Mackwitz, E Hesping, Y Antonova‐Koch, D Diedrich, ... ChemMedChem 14 (9), 912-926, 2019 | 28 | 2019 |
Artificial intelligence takes center stage: exploring the capabilities and implications of ChatGPT and other AI-assisted technologies in scientific research and education Immunology and Cell Biology 101 (10), 923-935, 2023 | 14 | 2023 |
Investigation of the in vitro and in vivo efficacy of peptoid-based HDAC inhibitors with dual-stage antiplasmodial activity MKW Mackwitz, E Hesping, K Eribez, A Schöler, Y Antonova-Koch, J Held, ... European Journal of Medicinal Chemistry 211, 113065, 2021 | 9 | 2021 |
QSAR Classification models for prediction of hydroxamate histone deacetylase inhibitor activity against malaria parasites E Hesping, MJ Chua, M Pflieger, Y Qian, L Dong, P Bachu, L Liu, T Kurz, ... ACS Infectious Diseases 8 (1), 106-117, 2022 | 5 | 2022 |
An ELISA method to assess HDAC inhibitor-induced alterations to P. falciparum histone lysine acetylation E Hesping, TS Skinner-Adams, GM Fisher, T Kurz, KT Andrews International Journal for Parasitology: Drugs and Drug Resistance 14, 249-256, 2020 | 5 | 2020 |
Histone deacetylase inhibitor AR-42 and achiral analogues kill malaria parasites in vitro and in mice MJ Chua, J Tng, E Hesping, GM Fisher, CD Goodman, T Skinner-Adams, ... International Journal for Parasitology: Drugs and Drug Resistance 17, 118-127, 2021 | 3 | 2021 |
MAM 2024: Malaria in a changing world RJ Longley, J Malinga, E Hesping, E Sutanto, SM DonVito, M Kucharski, ... Trends in Parasitology, 2024 | | 2024 |
Whole‐genome CRISPR screens to understand Apicomplexan–host interactions E Hesping, JA Boddey Molecular Microbiology, 2024 | | 2024 |
A broadly cross-reactive i-body to AMA1 potently inhibits blood and liver stages of Plasmodium parasites M Foley, D Angage, R Anders, J Chmielewski, J Maddumage, E Hesping, ... | | 2023 |
Genome-wide gene expression profiles throughout human malaria parasite liver stage development S Kappe, G Zanghi, H Patel, N Camargo, J Smith, Y Bae, E Hesping, ... | | 2023 |
A conserved malaria parasite protein required for maintenance of sporozoite cell shape and transmission JT Dessens, E Hesping Molecular microbiology 117 (6), 1293-1296, 2022 | | 2022 |
367 A targetable receptor-binding site on PfCyRPA to aid in the fight against malaria RJ Longley, J Malinga, E Hesping, E Sutanto, SM DonVito, M Kucharski, ... | | |