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Ludovica Monti
Ludovica Monti
Lecturer and Group Leader, The University of Melbourne
Verified email at unimelb.edu.au
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Cited by
Year
New indole tubulin assembly inhibitors cause stable arrest of mitotic progression, enhanced stimulation of natural killer cell cytotoxic activity, and repression of hedgehog …
G La Regina, R Bai, A Coluccia, V Famiglini, S Pelliccia, S Passacantilli, ...
Journal of medicinal chemistry 58 (15), 5789-5807, 2015
572015
Discovery of 1, 1′-biphenyl-4-sulfonamides as a new class of potent and selective carbonic anhydrase XIV inhibitors
G La Regina, A Coluccia, V Famiglini, S Pelliccia, L Monti, D Vullo, E Nuti, ...
Journal of medicinal chemistry 58 (21), 8564-8572, 2015
462015
Evaluation of oxetan-3-ol, thietan-3-ol, and derivatives thereof as bioisosteres of the carboxylic acid functional group
P Lassalas, K Oukoloff, V Makani, M James, V Tran, Y Yao, L Huang, ...
ACS Medicinal Chemistry Letters 8 (8), 864-868, 2017
452017
Multitargeted imidazoles: potential therapeutic leads for Alzheimer’s and other neurodegenerative diseases
AS Cornec, L Monti, J Kovalevich, V Makani, MJ James, KG Vijayendran, ...
Journal of medicinal chemistry 60 (12), 5120-5145, 2017
452017
Structure-Based Optimization of Quinazolines as Cruzain and TbrCATL Inhibitors
E Barbosa da Silva, DA Rocha, IS Fortes, W Yang, L Monti, ...
Journal of Medicinal Chemistry 64 (17), 13054-13071, 2021
282021
Brain‐penetrant triazolopyrimidine and phenylpyrimidine microtubule stabilizers as potential leads to treat human African trypanosomiasis
L Monti, SC Wang, K Oukoloff, AB Smith III, KR Brunden, CR Caffrey, ...
ChemMedChem 13 (17), 1751-1754, 2018
272018
Evaluation of the Structure–Activity Relationship of Microtubule-Targeting 1,2,4-Triazolo[1,5-a]pyrimidines Identifies New Candidates for Neurodegenerative …
K Oukoloff, G Nzou, C Varricchio, B Lucero, T Alle, J Kovalevich, L Monti, ...
Journal of medicinal chemistry 64 (2), 1073-1102, 2021
252021
Identification of anisomycin, prodigiosin and obatoclax as compounds with broad-spectrum anti-parasitic activity
G Ehrenkaufer, P Li, EE Stebbins, MM Kangussu-Marcolino, A Debnath, ...
PLoS neglected tropical diseases 14 (3), e0008150, 2020
222020
Long-range DNA interactions: Inter-molecular G-quadruplexes and their potential biological relevance
D Liano, L Monti, S Chowdhury, F Raguseo, M Di Antonio
Chemical Communications 58 (92), 12753-12762, 2022
192022
Arylboronic acids as dual-action FAAH and TRPV1 ligands
E Morera, V Di Marzo, L Monti, M Allarà, AS Moriello, M Nalli, G Ortar, ...
Bioorganic & Medicinal Chemistry Letters 26 (5), 1401-1405, 2016
152016
Evaluation of the analgesic effect of 4-anilidopiperidine scaffold containing ureas and carbamates
L Monti, A Stefanucci, S Pieretti, F Marzoli, L Fidanza, A Mollica, S Mirzaie, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (6), 1638-1647, 2016
122016
Drug Discovery and Development for Kinetoplastid Diseases
CR Caffrey, D Steverding, RS Ferreira, RB de Oliveira, AJ O'Donoghue, ...
Burger's Medicinal Chemistry and Drug Discovery, 8th Edition 7, 255-334, 2021
11*2021
Structure-activity relationship of dibenzylideneacetone analogs against the neglected disease pathogen, Trypanosoma brucei
KR Francisco, L Monti, W Yang, H Park, LJ Liu, K Watkins, ...
Bioorganic & medicinal chemistry letters 81, 129123, 2023
102023
Congeners Derived from Microtubule-Active Phenylpyrimidines Produce a Potent and Long-Lasting Paralysis of Schistosoma mansoni In Vitro
L Monti, AS Cornec, K Oukoloff, J Kovalevich, K Prijs, T Alle, KR Brunden, ...
ACS infectious diseases 7 (5), 1089-1103, 2020
92020
G-quadruplexes mark sites of methylation instability associated with ageing and cancer
J Rauchhaus, J Robinson, L Monti, M Di Antonio
Genes 13 (9), 1665, 2022
82022
From rational design to serendipity: discovery of novel thiosemicarbazones as potent trypanocidal compounds
SFP Braga, VC Santos, RP Vieira, EB da Silva, L Monti, SH Krake, ...
European Journal of Medicinal Chemistry 244, 114876, 2022
62022
Structure‐Activity Relationships, Tolerability and Efficacy of Microtubule‐Active 1,2,4‐Triazolo[1,5‐a]pyrimidines as Potential Candidates to Treat Human African …
L Monti, LJ Liu, C Varricchio, B Lucero, T Alle, W Yang, I Ben‐Shalom, ...
ChemMedChem 18 (20), e202300193, 2023
32023
G‐Quadruplexes as Key Transcriptional Regulators in Neglected Trypanosomatid Parasites
L Monti, M Di Antonio
ChemBioChem 24 (12), e202300265, 2023
32023
Front Cover: Structure‐Activity Relationships, Tolerability and Efficacy of Microtubule‐Active 1,2,4‐Triazolo[1,5‐a]pyrimidines as Potential Candidates to Treat …
L Monti, LJ Liu, C Varricchio, B Lucero, T Alle, W Yang, I Bem‐Shalom, ...
ChemMedChem 18 (20), e202300558, 2023
2023
Tubulin and Microtubules as Drug Targets for Potential Cancer Chemotherapy and CNS-Directed Therapies
L Monti
Sapienza Università Editrice, 2022
2022
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Articles 1–20