| Biomarker accessible and chemically addressable mechanistic subtypes of BRAF melanoma B Eskiocak, EA McMillan, S Mendiratta, RK Kollipara, H Zhang, ... Cancer discovery 7 (8), 832-851, 2017 | 60 | 2017 |
| Epigenetic profiling of the antitumor natural product psammaplin A and its analogues J García, G Franci, R Pereira, R Benedetti, A Nebbioso, ... Bioorganic & medicinal chemistry 19 (12), 3637-3649, 2011 | 58 | 2011 |
| Indole-derived psammaplin A analogues as epigenetic modulators with multiple inhibitory activities R Pereira, R Benedetti, S Perez-Rodriguez, A Nebbioso, ... Journal of Medicinal Chemistry 55 (22), 9467-9491, 2012 | 55 | 2012 |
| Death receptor pathway activation and increase of ROS production by the triple epigenetic inhibitor UVI5008 A Nebbioso, R Pereira, H Khanwalkar, F Matarese, J García-Rodríguez, ... Molecular cancer therapeutics 10 (12), 2394-2404, 2011 | 55 | 2011 |
| Diversity-oriented synthesis of diverse polycyclic scaffolds inspired by the logic of sesquiterpene lactones biosynthesis G lle Valot, JØ Garcia, V Duplan, C Serba, S Barluenga, N Winssinger | 45 | 2012 |
| Concise modular asymmetric synthesis of deguelin, tephrosin and investigation into their mode of action J Garcia, S Barluenga, K Beebe, L Neckers, N Winssinger Chemistry (Weinheim an der Bergstrasse, Germany) 16 (32), 9767, 2010 | 35 | 2010 |
| Synthesis of deguelin–biotin conjugates and investigation into deguelin’s interactions J Garcia, S Barluenga, K Gorska, F Sasse, N Winssinger Bioorganic & medicinal chemistry 20 (2), 672-680, 2012 | 25 | 2012 |
| Synthesis of sesquiterpene-inspired derivatives designed for covalent binding and their inhibition of the NF-κB pathway V Duplan, C Serba, J Garcia, G Valot, S Barluenga, M Hoerlé, M Cuendet, ... Organic & Biomolecular Chemistry 12 (2), 370-375, 2014 | 20 | 2014 |
| Pyrazine arotinoids with inverse agonist activities on the retinoid and rexinoid receptors J García, H Khanwalkar, R Pereira, C Erb, JJ Voegel, P Collette, ... ChemBioChem 10 (7), 1252-1259, 2009 | 18 | 2009 |
| Total synthesis of the natural isoprenylcysteine carboxyl methyltransferase inhibitor spermatinamine J García, R Pereira, AR de Lera Tetrahedron Letters 50 (35), 5028-5030, 2009 | 17 | 2009 |
| Synthesis and structure–activity studies of the V-ATPase inhibitor saliphenylhalamide (SaliPhe) and simplified analogs Jose Garcia-Rodriguez, Saurabh Mendiratta, Michael A. White, Xiao-Song Xie ... Bioorganic & Medicinal Chemistry Letters 25 (20), 4393-4398, 2015 | 16 | 2015 |
| Inhibition of IκB kinase-β and IκB kinase-α by heterocyclic adamantyl arotinoids J García-Rodríguez, S Pérez-Rodríguez, MA Ortiz, R Pereira, AR de Lera, ... Bioorganic & medicinal chemistry 22 (4), 1285-1302, 2014 | 9 | 2014 |
| SPOTLIGHTS... G Valot, J Garcia, V Duplan, C Serba, S Barluenga, N Winssinger | | |
