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| A Single‐Stranded DNA‐Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks G Bassi, N Favalli, M Vuk, M Catalano, A Martinelli, A Trenner, A Porro, ... Advanced Science 7 (22), 2001970, 2020 | 38 | 2020 |
| Chemical epigenetics: the impact of chemical and chemical biology techniques on bromodomain target validation M Schiedel, M Moroglu, DMH Ascough, AER Chamberlain, JJAG Kamps, ... Angewandte Chemie International Edition 58 (50), 17930-17952, 2019 | 29 | 2019 |
| BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability LE Jennings, M Schiedel, DS Hewings, S Picaud, CMC Laurin, PA Bruno, ... Bioorganic & Medicinal Chemistry 26 (11), 2937-2957, 2018 | 27 | 2018 |
| Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self‐assembly Chemical Library M Catalano, M Moroglu, P Balbi, F Mazzieri, J Clayton, KH Andrews, ... ChemMedChem 15 (18), 1752-1756, 2020 | 19 | 2020 |
| Controlling intramolecular interactions in the design of selective, high-affinity ligands for the CREBBP bromodomain M Brand, J Clayton, M Moroglu, M Schiedel, S Picaud, JP Bluck, ... Journal of medicinal chemistry 64 (14), 10102-10123, 2021 | 16 | 2021 |
| Chemische Epigenetik: der Einfluss chemischer und chemo‐biologischer Techniken auf die Zielstruktur‐Validierung von Bromodomänen M Schiedel, M Moroglu, DMH Ascough, AER Chamberlain, JJAG Kamps, ... Angewandte Chemie 131 (50), 18096-18120, 2019 | 2 | 2019 |
| Controlling Intramolecular Interactions in the Design of Selective, High-Affinity, Ligands for the CREBBP Bromodomain (preprint) M Brand, J Clayton, M Moroglu, M Schiedel, S Picaud, J Bluck, ... | | 2020 |
| Development of small molecule CREBBP bromodomain ligands using medicinal chemistry-based approaches M Moroglu University of Oxford, 2020 | | 2020 |
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