| Lithium enolates in the enantioselective construction of tetrasubstituted carbon centers with chiral lithium amides as noncovalent stereodirecting auxiliaries K Yu, P Lu, JJ Jackson, TAD Nguyen, J Alvarado, CE Stivala, Y Ma, ... Journal of the American Chemical Society 139 (1), 527-533, 2017 | 55 | 2017 |
| Stereoselective synthesis of 1, 3-amino alcohols by the Pd-catalyzed cyclization of trichloroacetimidates Y Xie, K Yu, Z Gu The Journal of Organic Chemistry 79 (3), 1289-1302, 2014 | 32 | 2014 |
| Direct enantioselective and regioselective alkylation of β, γ-unsaturated carboxylic acids with chiral lithium amides as traceless auxiliaries K Yu, B Miao, W Wang, A Zakarian Organic letters 21 (6), 1930-1934, 2019 | 22 | 2019 |
| N-Bromoacetamide-mediated domino cyclization and elimination of homoallylic trichloroacetimidates: a novel approach toward the synthesis of 1-bromo-2-amino-3-butene derivatives R Zhu, K Yu, Z Gu Organic & Biomolecular Chemistry 12 (34), 6653-6660, 2014 | 5 | 2014 |
| 46P AB521, a clinical-stage, potent, and selective Hypoxia-Inducible Factor (HIF)-2α inhibitor, for the treatment of renal cell carcinoma KV Lawson, KES Gauthier, D Piovesan, A Mailyan, G Mata, JTA Fournier, ... Annals of Oncology 33, S21, 2022 | 2 | 2022 |
| Abstract P206: AB521 potently and selectively inhibits pro-tumorigenic gene transcription by Hypoxia-Inducible Factor (HIF)-2α in vitro and in vivo KES Gauthier, D Piovesan, S Cho, KV Lawson, PG Schweickert, A Lopez, ... Molecular Cancer Therapeutics 20 (12_Supplement), P206-P206, 2021 | 1 | 2021 |
| TETRALIN AND TETRAHYDROQUINOLINE COMPOUNDS AS INHIBITORS OF HIF-2ALPHA JW Beatty, SL Drew, M Epplin, JTA Fournier, B Gal, T Guney, KT Haelsig, ... WO Patent WO2021/188,769, 2021 | 1 | 2021 |
| Cbl inhibition increases the response of cytotoxic T cells to sub-optimal stimulation and drives enhanced anti-tumor responses alone or in combination with PD-1 blockade L Yamashiro, S Marubayashi, R Rayaji, A Battsooj, K Mrouj, H Singh, ... Cancer Research 84 (6_Supplement), 4042-4042, 2024 | | 2024 |
| Cbl-b inhibitors and methods of use thereof JW Beatty, B Gal, SK Gangam, C Hardman, MR Leleti, KV Lawson, D Liu, ... WO Patent WO2024020034A1, 2023 | | 2023 |
| Inhibitors of hif-2alpha and methods of use thereof JW Beatty, SL Drew, M Epplin, J Fournier, GAL Balint, C Hardman, ... US Patent App. 18/050,557, 2023 | | 2023 |
| SUBSTITUTED PYRROLO [2, 3-b] PYRIDINE AND PYRAZOLO [3, 4-b] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS H TAN, Q LIU, B LIU, Z LI, X WANG, Z ZHOU, W ZHANG, Y WANG, ... WO Patent WO 2020/239124 A1, 2020 | | 2020 |
Thuy-Ai D. NguyenScientist, Los Alamos National LabVerified email at lanl.gov
