Methods to identify and optimize small molecules interacting with RNA (SMIRNAs) A Ursu, S Vézina-Dawod, MD Disney Drug Discovery Today 24 (10), 2002-2016, 2019 | 30 | 2019 |
DNA-encoded library versus RNA-encoded library selection enables design of an oncogenic noncoding RNA inhibitor RI Benhamou, BM Suresh, Y Tong, WG Cochrane, V Cavett, ... Proceedings of the National Academy of Sciences 119 (6), e2114971119, 2022 | 29 | 2022 |
Convenient two-step synthesis of highly functionalized benzo-fused 1, 4-diazepin-3-ones and 1, 5-diazocin-4-ones by sequential Ugi and intramolecular SNAr reactions S Vezina-Dawod, N Gerber, X Liang, E Biron Tetrahedron 73 (44), 6347-6355, 2017 | 22 | 2017 |
Preparation of N-Substituted N-Arylsulfonylglycines and Their Use in Peptoid Synthesis S Jobin, S Vezina-Dawod, C Herby, A Derson, E Biron Organic letters 17 (22), 5626-5629, 2015 | 16 | 2015 |
One-pot photochemical ring-opening/cleavage approach for the synthesis and decoding of cyclic peptide libraries X Liang, S Vézina-Dawod, F Bédard, K Porte, E Biron Organic letters 18 (5), 1174-1177, 2016 | 14 | 2016 |
N-substituted arylsulfonamide building blocks as alternative submonomers for peptoid synthesis S Vézina-Dawod, A Derson, E Biron Tetrahedron letters 56 (2), 382-385, 2015 | 13 | 2015 |
Toward solid-phase peptide fragment ligation by a traceless-Ugi multicomponent reaction approach S Jobin, A Méjean, SM Galindo, X Liang, S Vézina-Dawod, E Biron Organic & Biomolecular Chemistry 14 (47), 11230-11237, 2016 | 12 | 2016 |
Massively parallel optimization of the linker domain in small molecule dimers targeting a toxic r (CUG) repeat expansion S Vezina-Dawod, AJ Angelbello, S Choudhary, KW Wang, I Yildirim, ... ACS Medicinal Chemistry Letters 12 (6), 907-914, 2021 | 6 | 2021 |
Synthetic strategies for macrocyclic peptides É Biron, S Vézina‐Dawod, F Bédard Practical Medicinal Chemistry with Macrocycles: Design, Synthesis, and Case …, 2017 | 6 | 2017 |
Macrocyclization of a ligand targeting a toxic RNA dramatically improves potency RI Benhamou, S Vezina‐Dawod, S Choudhary, K Won Wang, SM Meyer, ... ChemBioChem 21 (22), 3229-3233, 2020 | 4 | 2020 |
Synthesis and biological evaluation of novel 1, 4-benzodiazepin-3-one derivatives as potential antitumor agents against prostate cancer S Vezina-Dawod, M Perreault, LD Guay, N Gerber, S Gobeil, E Biron Bioorganic & Medicinal Chemistry 45, 116314, 2021 | 3 | 2021 |
Design, synthèse et criblage de chimiothèques peptidomimétiques pour la découverte d'agents antinéoplasiques S Vézina-Dawod PhD's thesis, 2018 | 1 | 2018 |
Synthesis and biological evaluation of novel 1, 4-benzodiazepin-3-one derivatives as potential antitumor agents against prostate cancer É Biron, S Gobeil, S Vézina-Dawod, N Gerber, LD Guay, M Perreault Pergamon, 2021 | | 2021 |
Convenient two-step synthesis of highly functionalized benzo-fused 1, 4-diazepin-3-ones and 1, 5-diazocin-4-ones by sequential Ugi and intramolecular SNAr reactions É Biron, S Vézina-Dawod, X Liang, N Gerber Pergamon Press, 2017 | | 2017 |
Toward solid-phase peptide fragment ligation by a traceless-Ugi multicomponent approach S Jobin, A Méjean, SM Galindo, X Liang, S Vézina-Dawod, E Biron Application de la réaction multicomposante de Ugi à la synthèse de peptides …, 2017 | | 2017 |
Preparation of N-substituted N-arylsulfonylglycines and their use in peptoid synthesis É Biron, S Jobin, C Herby, S Vézina-Dawod, A Derson American Chemical Society, 2015 | | 2015 |
N-Substituted arylsulfonamide building blocks as alternative submonomers for peptoid synthesis É Biron, A Derson, S Vézina-Dawod Elsevier, 2015 | | 2015 |
Towards the Development of Cell Permeable Macrocyclic Scaffolds: Probing the Structural Requirements for Enhancing Cellular Uptake S Vézina-Dawod, S Fortin, M Perrin, LJ Bordeleau, S Gobeil, E Biron Peptide 2015: Proceedings of the 24th American Peptide Symposium, 127-130, 2015 | | 2015 |
Design et synthèse de macrocycles pseudopeptidiques pour le développement d'inhibiteurs d'interactions protéine-protéine S Vézina-Dawod Master's thesis, 2015 | | 2015 |
N-Substituted Arylsulfonamides as Alternative Building Blocks in Peptoid and Peptide Synthesis S Vézina-Dawod, S Jobin, A Derson, C Herby, E Biron Peptide 2015: Proceedings of the 24th American Peptide Symposium, 280-282, 2015 | | 2015 |