| 3CL protease inhibitors with an electrophilic arylketone moiety as anti-SARS-CoV-2 agents S Konno, K Kobayashi, M Senda, Y Funai, Y Seki, I Tamai, L Schäkel, ... Journal of Medicinal Chemistry 65 (4), 2926-2939, 2021 | 109 | 2021 |
| Development of potent dipeptide-type SARS-CoV 3CL protease inhibitors with novel P3 scaffolds: design, synthesis, biological evaluation, and docking studies P Thanigaimalai, S Konno, T Yamamoto, Y Koiwai, A Taguchi, ... European journal of medicinal chemistry 68, 372-384, 2013 | 104 | 2013 |
| Design and synthesis of new tripeptide-type SARS-CoV 3CL protease inhibitors containing an electrophilic arylketone moiety S Konno, P Thanigaimalai, T Yamamoto, K Nakada, R Kakiuchi, ... Bioorganic & medicinal chemistry 21 (2), 412-424, 2013 | 79 | 2013 |
| Design, synthesis, and biological evaluation of novel dipeptide-type SARS-CoV 3CL protease inhibitors: Structure–activity relationship study P Thanigaimalai, S Konno, T Yamamoto, Y Koiwai, A Taguchi, ... European journal of medicinal chemistry 65, 436-447, 2013 | 78 | 2013 |
| Active site-directed proteomic probes for adenylation domains in nonribosomal peptide synthetases S Konno, F Ishikawa, T Suzuki, N Dohmae, MD Burkart, H Kakeya Chemical communications 51 (12), 2262-2265, 2015 | 34 | 2015 |
| Accurate detection of Adenylation domain functions in nonribosomal peptide Synthetases by an enzyme-linked immunosorbent assay system using active site-directed probes for … F Ishikawa, K Miyamoto, S Konno, S Kasai, H Kakeya ACS Chemical Biology 10 (12), 2816-2826, 2015 | 23 | 2015 |
| Profiling nonribosomal peptide synthetase activities using chemical proteomic probes for adenylation domains F Ishikawa, S Konno, T Suzuki, N Dohmae, H Kakeya ACS Chemical Biology 10 (9), 1989-1997, 2015 | 23 | 2015 |
| Functional profiling of adenylation domains in nonribosomal peptide synthetases by competitive activity-based protein profiling S Kasai, S Konno, F Ishikawa, H Kakeya Chemical communications 51 (87), 15764-15767, 2015 | 21 | 2015 |
| Chemoproteomics profiling of surfactin-producing nonribosomal peptide synthetases in living bacterial cells F Ishikawa, S Konno, C Uchida, T Suzuki, K Takashima, N Dohmae, ... Cell Chemical Biology 29 (1), 145-156. e8, 2022 | 16 | 2022 |
| Trapping the complex molecular machinery of polyketide and fatty acid synthases with tunable silylcyanohydrin crosslinkers S Konno, JJ La Clair, MD Burkart Angewandte Chemie 130 (52), 17255-17259, 2018 | 13 | 2018 |
| Structural revision of natural cyclic depsipeptide MA026 established by total synthesis and biosynthetic gene cluster analysis C Uchiyama, A Fukuda, M Mukaiyama, Y Nakazawa, Y Kuramochi, ... Angewandte Chemie International Edition 60 (16), 8792-8797, 2021 | 7 | 2021 |
| Exploring a chemical scaffold for rapid and selective photoaffinity labelling of non-ribosomal peptide synthetases in living bacterial cells F Ishikawa, S Konno, Y Uchiyama, H Kakeya, G Tanabe Philosophical Transactions of the Royal Society B 378 (1871), 20220026, 2023 | 4 | 2023 |
| Chemical Synthesis of an HIV-1 Protease Analog with Some Amides in a Polypeptide Main Chain Replaced by Disulfide Bonds Y Cui, A Taguchi, H Shida, S Konno, K Takayama, A Taniguchi, ... Bulletin of the Chemical Society of Japan 95 (8), 1156-1162, 2022 | 3 | 2022 |
| Inhibition of efflux pumps aids small-molecule probe-based fluorescence labeling and imaging in the Gram-negative bacterium Escherichia coli F Ishikawa, S Konno, K Takashima, H Kakeya, G Tanabe Organic & Biomolecular Chemistry 19 (41), 8906-8911, 2021 | 3 | 2021 |
| Development of functionalized peptides for efficient inhibition of myostatin by selective photooxygenation H Okamoto, A Taniguchi, S Usami, M Katsuyama, S Konno, A Taguchi, ... Organic & Biomolecular Chemistry 19 (1), 199-207, 2021 | 3 | 2021 |
| A chemoproteomics approach to investigate phosphopantetheine transferase activity at the cellular level S Konno, F Ishikawa, T Suzuki, N Dohmae, H Kakeya, G Tanabe ChemBioChem 18 (18), 1855-1862, 2017 | 3 | 2017 |
| Establishment of One-Pot Disulfide-Driven Cyclic Peptide Synthesis with a 3-Nitro-2-pyridinesulfenate H Shida, A Taguchi, S Konno, K Takayama, A Taniguchi, Y Hayashi Chemical and Pharmaceutical Bulletin 71 (6), 435-440, 2023 | 1 | 2023 |
| In silico design of inhibitor against SARS-CoV-2 protease by docking simulation and ADMET prediction M Hoshi, S Shiino, A Gomi, K Sakata, S Konno, Y Hayashi, M Kojima bioimages 29, 11-21, 2021 | 1 | 2021 |
| Thioesterase domain-mediated macrocyclization of non-ribosomal peptides S Konno, L Misson, MD Burkart | 1 | 2017 |
| Detection of Active SARS-CoV-2 3CL Protease in Infected Cells Using Activity-Based Probes with a 2, 6-Dichlorobenzoyloxymethyl Ketone Reactive Warhead Y Yamauchi, S Konno, N Omura, N Yoshioka, A Hingst, M Gütschow, ... ACS Chemical Biology, 2024 | | 2024 |
