Small molecule inhibitors of bromodomain–acetyl-lysine interactions M Brand, AM Measures, BG Wilson, WA Cortopassi, R Alexander, ... ACS chemical biology 10 (1), 22-39, 2014 | 163 | 2014 |
Chemical epigenetics: the Impact of chemical and chemical biology techniques on bromodomain target validation M Schiedel, M Moroglu, DMH Ascough, AER Chamberlain, JJAG Kamps, ... Angewandte Chemie International Edition 58 (50), 17930-17952, 2019 | 29 | 2019 |
Isoxazole‐Derived Amino Acids are Bromodomain‐Binding Acetyl‐Lysine Mimics: Incorporation into Histone H4 Peptides and Histone H3 AR Sekirnik, DS Hewings, NH Theodoulou, L Jursins, KR Lewendon, ... Angewandte Chemie International Edition 55 (29), 8353-8357, 2016 | 27 | 2016 |
Structure–activity relationships and colorimetric properties of specific probes for the putative cancer biomarker human arylamine N-acetyltransferase 1 JE Egleton, CC Thinnes, PT Seden, N Laurieri, SP Lee, KS Hadavizadeh, ... Bioorganic & medicinal chemistry 22 (11), 3030-3054, 2014 | 27 | 2014 |
Phenotypic screening and fragment-based approaches to the discovery of small-molecule bromodomain ligands LE Jennings, AR Measures, BG Wilson, SJ Conway Future medicinal chemistry 6 (2), 179-204, 2014 | 19 | 2014 |
Chemische Epigenetik: der Einfluss chemischer und chemo‐biologischer Techniken auf die Zielstruktur‐Validierung von Bromodomänen M Schiedel, M Moroglu, DMH Ascough, AER Chamberlain, JJAG Kamps, ... Angewandte Chemie 131 (50), 18096-18120, 2019 | 2 | 2019 |