| Design, multigram synthesis, and in vitro and in vivo evaluation of propylamycin: A semisynthetic 4, 5-deoxystreptamine class aminoglycoside for the treatment of drug-resistant … T Matsushita, GC Sati, N Kondasinghe, MG Pirrone, T Kato, P Waduge, ... Journal of the American Chemical Society 141 (12), 5051-5061, 2019 | 57 | 2019 |
| Fluoride migration catalysis enables simple, stereoselective, and iterative glycosylation GC Sati, JL Martin, Y Xu, T Malakar, PM Zimmerman, J Montgomery Journal of the American Chemical Society 142 (15), 7235-7242, 2020 | 50 | 2020 |
| Modification at the 2′-position of the 4, 5-series of 2-deoxystreptamine aminoglycoside antibiotics to resist aminoglycoside modifying enzymes and increase ribosomal target … GC Sati, VA Sarpe, T Furukawa, S Mondal, M Mantovani, SN Hobbie, ... ACS infectious diseases 5 (10), 1718-1730, 2019 | 32 | 2019 |
| Assessing the role of dopamine in the differential neurotoxicity patterns of methamphetamine, mephedrone, methcathinone and 4-methylmethamphetamine JH Anneken, M Angoa-Perez, GC Sati, D Crich, DM Kuhn Neuropharmacology 134, 46-56, 2018 | 29 | 2018 |
| Dissecting the influence of two structural substituents on the differential neurotoxic effects of acute methamphetamine and mephedrone treatment on dopamine nerve endings with … JH Anneken, M Angoa-Pérez, GC Sati, D Crich, DM Kuhn Journal of Pharmacology and Experimental Therapeutics 360 (3), 417-423, 2017 | 21 | 2017 |
| N6′, N6′′′, and O4′ modifications to neomycin affect ribosomal selectivity without compromising antibacterial activity GC Sati, D Shcherbakov, SN Hobbie, A Vasella, EC Bottger, D Crich ACS infectious diseases 3 (5), 368-377, 2017 | 16 | 2017 |
| Facile Synthesis of 3-N-Alkyl Pyrimidin-2,4-diones from N-Sulfonyloxy Maleimides and Amines GC Sati, D Crich Organic letters 17 (16), 4122-4124, 2015 | 15 | 2015 |
| Structure‐Activity Relationships for 5′′ Modifications of 4, 5‐Aminoglycoside Antibiotics JCK Quirke, GC Sati, A Sonousi, M Gysin, K Haldimann, EC Böttger, ... ChemMedChem 17 (13), e202200120, 2022 | 10 | 2022 |
| Synthesis and Antibacterial Activity of Propylamycin Derivatives Functionalized at the 5′′-and Other Positions with a View to Overcoming Resistance Due to Aminoglycoside … D Lubriks, R Zogota, VA Sarpe, T Matsushita, GC Sati, K Haldimann, ... ACS infectious diseases 7 (8), 2413-2424, 2021 | 10 | 2021 |
| 2. The Exploration of Aza-quinolines as Hematopoietic Prostaglandin D Synthase (H-PGDS) Inhibitors with Low Brain Exposure. Bioorg. Med. Chem. 28 (23), 115791, 2020 | 6 | 2020 |
| Use of a fluorescence assay to determine relative affinities of semisynthetic aminoglycosides to small RNAs representing bacterial and mitochondrial A sites P Waduge, GC Sati, D Crich, CS Chow Bioorganic & medicinal chemistry 27 (22), 115121, 2019 | 6 | 2019 |
| Dissociation between hypothermia and neurotoxicity caused by mephedrone and methcathinone in TPH2 knockout mice JH Anneken, M Angoa-Perez, GC Sati, D Crich, DM Kuhn Psychopharmacology 236, 1097-1106, 2019 | 6 | 2019 |
| Glycosyl Exchange of Unactivated Glycosidic Bonds: Suppressing or Embracing Side Reactivity in Catalytic Glycosylations JM Joshua L. Martin, Girish C. Sati, Tanmay Malakar, Jessica Hatt, Paul M ... The Journal of Organic Chemistry 87 (9), 5817–5826, 2022 | 4 | 2022 |
| Copper-Catalyzed Intermolecular Thioamination of Maleimides with Thiols and Formamides: A One-Step Construction of 3-Amino-4-thiomaleimides Using Formamides as Nitrogen Sources ZH Yang, JN Zhu, ZH Jin, J Zheng, SY Zhao Synthesis 50 (23), 4627-4636, 2018 | 4 | 2018 |
| Addressing The Threat Of Multidrug Resistant Infectious Diseases By Synthesis Of Novel Aminoglycoside Antibiotics GC Sati | 1 | 2018 |
| Neomycin and paromomycin derivatives D Crich, S Girish, A Sonousi, G Yang, AR Mandhapati, MG Pirrone, T Kato, ... US Patent 11,466,044, 2022 | | 2022 |
| Methods for Glycosylation J Montgomery, GC Sati, JL Martin US Patent App. 17/610,996, 2022 | | 2022 |
| Design, synthesis, and evaluation of improved aminoglycosides M Pirrone, T Matsushita, G Sati, T Kato, S Hobbie, T Schrepfer, J Schacht, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 256, 2018 | | 2018 |
| Dissecting the influence of two structural substituents on the differential neurotoxic effects of methamphetamine and mephedrone on dopamine nerve endings with the use of 4 … JH Anneken, M Angoa-Perez, GC Sati, D Crich, DM Kuhn Journal of Pharmacology and Experimental Therapeutics, 2016 | | 2016 |
| Concise synthesis of highly functionalized pyrimidine-2, 4-(1H, 3H)-dione derivatives G Sati, D Crich, E Bottger, A Vasella ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 250, 2015 | | 2015 |
Michael G PirronePost Doctoral Associate, University of GeorgiaVerified email at uga.edu
