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Eric A. Wold
Eric A. Wold
U.S. Naval Research Laboratory
Verified email at rice.edu - Homepage
Title
Cited by
Cited by
Year
Therapeutic Potential of Spirooxindoles as Antiviral Agents
N Ye, H Chen, EA Wold, PY Shi, J Zhou
ACS Infectious Diseases 2 (6), 382-392, 2016
3742016
Drug Discovery Targeting Bromodomain-Containing Protein 4
Z Liu, P Wang, H Chen, EA Wold, B Tian, AR Brasier, J Zhou
Journal of Medicinal Chemistry 60 (11), 4533-4558, 2017
2692017
Discovery and development of natural product oridonin-inspired anticancer agents
Y Ding, C Ding, N Ye, Z Liu, EA Wold, H Chen, C Wild, Q Shen, J Zhou
European Journal of Medicinal Chemistry 122, 102-117, 2016
1642016
Allosteric Modulation of Class A GPCRs: Targets, Agents, and Emerging Concepts
EA Wold, J Chen, KA Cunningham, J Zhou
Journal of Medicinal Chemistry 62 (1), 88-127, 2018
1412018
Therapeutic Potential of Oridonin and Its Analogs: From Anticancer and Antiinflammation to Neuroprotection
J Xu, EA Wold, Y Ding, Q Shen, J Zhou
Molecules 23 (2), 474, 2018
1082018
BH4 domain of Bcl-2 as a novel target for cancer therapy
Z Liu, C Wild, Y Ding, N Ye, H Chen, EA Wold, J Zhou
Drug Discovery Today 21 (6), 989-996, 2016
642016
Discovery of Orally Bioavailable Chromone Derivatives as Potent and Selective BRD4 Inhibitors: Scaffolding Hopping, Optimization and Pharmacological Evaluation
Z Liu, H Chen, P Wang, Y Li, EA Wold, PG Leonard, S Joseph, AR Brasier, ...
Journal of Medicinal Chemistry 63 (10), 5242-5256, 2020
612020
Small Molecules Selectively Targeting Sigma-1 Receptor for the Treatment of Neurological Diseases
N Ye, W Qin, S Tian, Q Xu, EA Wold, J Zhou, XC Zhen
Journal of Medicinal Chemistry 63 (24), 15187-15217, 2020
602020
Targeting the 5-HT2C Receptor in Biological Context and the Current State of 5-HT2C Receptor Ligand Development.
EA Wold, CT Wild, KA Cunningham, J Zhou
Current Topics in Medicinal Chemistry 19, 1381-1398, 2019
482019
Regio-and Stereospecific Synthesis of Oridonin D-Ring Aziridinated Analogues for the Treatment of Triple-Negative Breast Cancer via Mediated Irreversible Covalent Warheads
Y Ding, D Li, C Ding, P Wang, Z Liu, EA Wold, N Ye, H Chen, MA White, ...
Journal of Medicinal Chemistry 61 (7), 2737-2752, 2018
332018
Design, Synthesis, and Characterization of 4-Undecylpiperidine-2-Carboxamides as Positive Allosteric Modulators of the Serotonin (5-HT) 5-HT2C Receptor
CT Wild, JM Miszkiel, EA Wold, CA Soto, C Ding, RM Hartley, MA White, ...
Journal of Medicinal Chemistry 62 (1), 288-305, 2018
312018
Orphan Receptor GPR88 as an Emerging Neurotherapeutic Target
N Ye, B Li, Q Mao, EA Wold, S Tian, JA Allen, J Zhou
ACS Chemical Neuroscience 10 (1), 190-200, 2019
302019
Small-Molecule Inhibitors Targeting the Canonical WNT Signaling Pathway for the Treatment of Cancer
Z Liu, P Wang, EA Wold, Q Song, C Zhao, C Wang, J Zhou
Journal of Medicinal Chemistry 64 (8), 4257-4288, 2021
282021
Discovery, X-ray Crystallography, and Anti-inflammatory Activity of Bromodomain-containing Protein 4 (BRD4) BD1 Inhibitors Targeting a Distinct New Binding Site
Z Liu, Y Li, H Chen, H Lai, P Wang, S Wu, EA Wold, PG Leonard, ...
Journal of Medicinal Chemistry 65 (3), 2388-2408, 2022
262022
GPCR Allosteric Modulators: Mechanistic Advantages and Therapeutic Applications
EA Wold, J Zhou
Current Topics in Medicinal Chemistry 18 (23), 2002-2006, 2019
262019
Inorganic arsenic–related changes in the stromal tumor microenvironment in a prostate cancer cell–conditioned media model
JJ Shearer, EA Wold, CS Umbaugh, CF Lichti, CL Nilsson, ML Figueiredo
Environmental Health Perspectives 124 (7), 1009, 2016
222016
Discovery of 4-Phenylpiperidine-2-Carboxamide Analogues as Serotonin 5-HT2C Receptor Positive Allosteric Modulators with Enhanced Drug-Like Properties
EA Wold, EJ Garcia, CT Wild, JM Miszkiel, CA Soto, J Chen, K Pazdrak, ...
Journal of Medicinal Chemistry 63 (14), 7529-7544, 2020
182020
Small-Molecule Inhibitors of Protein-Protein Interactions
Z Liu, H Chen, EA Wold, J Zhou
Reference Module in Chemistry, Molecular Sciences and Chemical Engineering …, 2017
142017
Structure-Activity Relationship Studies on Bax Activator SMBA1 for the Treatment of ER-Positive and Triple-Negative Breast Cancer
G Liu, T Yin, H Kim, C Ding, Z Yu, H Wang, H Chen, R Yan, EA Wold, ...
European Journal of Medicinal Chemistry 178, 589-605, 2019
132019
Applications of Bioorthogonal Chemistry in Tumor-Targeted Drug Discovery
G Liu, EA Wold, J Zhou
Current Topics in Medicinal Chemistry 19 (11), 892-897, 2019
122019
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