Small molecule modulation of the Drosophila Slo channel elucidated by cryo-EM T Raisch, A Brockmann, U Ebbinghaus-Kintscher, J Freigang, O Gutbrod, ... Nature communications 12 (1), 7164, 2021 | 14 | 2021 |
Towards understanding transfluthrin efficacy in a pyrethroid-resistant strain of the malaria vector Anopheles funestus with special reference to cytochrome P450-mediated … M Nolden, A Brockmann, U Ebbinghaus-Kintscher, KU Brueggen, ... Current Research in Parasitology & Vector-borne Diseases 1, 100041, 2021 | 14 | 2021 |
Cryo-EM structural studies of the agonist complexed human TRPV4 ion-channel reveals novel structural rearrangements resulting in an open-conformation M Botte, AKC Ulrich, R Adaixo, D Gnutt, A Brockmann, D Bucher, ... BioRxiv, 2020.10. 13.334797, 2020 | 14 | 2020 |
Novel, dual target‐directed annelated xanthine derivatives acting on adenosine receptors and monoamine oxidase B KJ Kuder, M Załuski, J Schabikowski, G Latacz, A Olejarz‐Maciej, P Jaśko, ... ChemMedChem 15 (9), 772-786, 2020 | 10 | 2020 |
8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation M Załuski, J Schabikowski, P Jaśko, A Bryła, A Olejarz-Maciej, M Kaleta, ... Bioorganic Chemistry 101, 104033, 2020 | 7 | 2020 |
Cryo-EM structural studies of the agonist complexed human TRPV4 ion-channel reveals novel structural rearrangements resulting in an open-conformation. bioRxiv: 2020.2010. 2013 … M Botte, AKC Ulrich, R Adaixo, D Gnutt, A Brockmann, D Bucher, ... | 5 | 2020 |
Anti-Inflammatory Activities of 8-Benzylaminoxanthines Showing High Adenosine A2A and Dual A1/A2A Receptor Affinity M Załuski, D Łażewska, P Jaśko, E Honkisz-Orzechowska, KJ Kuder, ... International Journal of Molecular Sciences 24 (18), 13707, 2023 | 2 | 2023 |
Implementation of a high throughput screening assay to identify and characterize insecticides acting on ion channels A Brockmann Universitäts-und Landesbibliothek Bonn, 2023 | | 2023 |
Characterization of Drosophila melanogaster slo1 channel using mutagenesis and automated patch clamp measurements on syncropatch384 (nanion technologies) A Brockmann, U Ebbinghaus-Kintscher Biophysical Journal 121 (3), 389a, 2022 | | 2022 |
8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A (2A) receptors. Design, synthesis and biological evaluation M Zaluski, J Schabikowski, P Jasko, A Bryla, A Olejarz-Maciej, M Kaleta, ... BIOORGANIC CHEMISTRY 101, 2020 | | 2020 |