Discovery of nonpungent transient receptor potential vanilloid 1 (TRPV1) agonist as strong topical analgesic J Ann, HS Kim, SA Thorat, H Kim, HJ Ha, K Choi, YH Kim, M Kim, ... Journal of medicinal chemistry 63 (1), 418-424, 2019 | 37 | 2019 |
Multi-functional diarylurea small molecule inhibitors of TRPV1 with therapeutic potential for neuroinflammation Z Feng, LV Pearce, Y Zhang, C Xing, BKA Herold, S Ma, Z Hu, NA Turcios, ... The AAPS journal 18, 898-913, 2016 | 24 | 2016 |
Discovery of benzopyridone-based transient receptor potential vanilloid 1 agonists and antagonists and the structural elucidation of their activity shift SA Thorat, Y Lee, A Jung, J Ann, S Ahn, J Baek, D Zuo, N Do, JJ Jeong, ... Journal of Medicinal Chemistry 64 (1), 370-384, 2021 | 13 | 2021 |
2-Sulfonamidopyridine C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl) propanamides as potent TRPV1 antagonists J Ann, Y Ki, S Yoon, MS Kim, JU Lee, C Kim, S Lee, A Jung, J Baek, ... Bioorganic & medicinal chemistry 24 (6), 1231-1240, 2016 | 12 | 2016 |
Discovery of N-(3-fluoro-4-methylsulfonamidomethylphenyl) urea as a potent TRPV1 antagonistic template J Ann, W Sun, X Zhou, A Jung, J Baek, S Lee, C Kim, S Yoon, S Hong, ... Bioorganic & medicinal chemistry letters 26 (15), 3603-3607, 2016 | 10 | 2016 |