The Chemogenetic Receptor Ligand Clozapine N-Oxide Induces in vivo Neuroreceptor Occupancy and Reduces Striatal Glutamate Levels S Bærentzen, A Casado-Sainz, D Lange, V Shalgunov, IM Tejada, ... Frontiers in Neuroscience 13, 187, 2019 | 41 | 2019 |
Improved radiosynthesis and preliminary in vivo evaluation of the 11C-labeled tetrazine [11C] AE-1 for pretargeted PET imaging EJL Stéen, JT Jørgensen, IN Petersen, K Nørregaard, S Lehel, ... Bioorganic & Medicinal Chemistry Letters 29 (8), 986-990, 2019 | 22 | 2019 |
In Vivo Veritas: 18F-Radiolabeled Glycomimetics Allow Insights into the Pharmacological Fate of Galectin-3 Inhibitors K Bratteby, E Torkelsson, ET L’Estrade, K Peterson, V Shalgunov, ... Journal of Medicinal Chemistry 63 (2), 747-755, 2019 | 21 | 2019 |
Towards selective CNS PET imaging of the 5-HT7 receptor system: Past, present and future ET L'Estrade, M Erlandsson, FG Edgar, T Ohlsson, GM Knudsen, ... Neuropharmacology 172, 107830, 2020 | 20 | 2020 |
Quantification accuracy of a new HRRT high throughput rat hotel using transmission-based attenuation correction: a phantom study SH Keller, EN L'Estrade, B Dall, M Palner, M Herth 2016 IEEE Nuclear Science Symposium, Medical Imaging Conference and Room …, 2016 | 16 | 2016 |
Classics in neuroimaging: the serotonergic 2A receptor system—from discovery to modern molecular imaging E T. L’Estrade, HD Hansen, M Erlandsson, TG Ohlsson, GM Knudsen, ... ACS Chemical Neuroscience 9 (6), 1226-1229, 2018 | 14 | 2018 |
Blocking of efflux transporters in rats improves translational validation of brain radioligands V Shalgunov, M Xiong, ET L’Estrade, NR Raval, IV Andersen, FG Edgar, ... EJNMMI research 10, 1-11, 2020 | 12 | 2020 |
Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of [18F]ENL30: A Potential PET Radiotracer for the 5-HT7 Receptor E Tampio L’Estrade, FG Edgar, M Xiong, V Shalgunov, SL Baerentzen, ... ACS omega 4 (4), 7344-7353, 2019 | 11 | 2019 |
The α-synuclein PET tracer [18F] ACI-12589 distinguishes multiple system atrophy from other neurodegenerative diseases R Smith, F Capotosti, M Schain, T Ohlsson, E Vokali, J Molette, ... Nature communications 14 (1), 6750, 2023 | 9 | 2023 |
In Vitro and In Vivo Characterization of Dibenzothiophene Derivatives [125I]Iodo-ASEM and [18F]ASEM as Radiotracers of Homo- and Heteromeric α7 Nicotinic … CK Donat, HH Hansen, HD Hansen, RC Mease, AG Horti, MG Pomper, ... Molecules 25 (6), 1425, 2020 | 9 | 2020 |
Development and Evaluation of Two Potential 5-HT7 Receptor PET Tracers: [18F]ENL09 and [18F]ENL10 E Tampio L’Estrade, M Xiong, V Shalgunov, FG Edgar, B Volk, ... ACS Chemical Neuroscience 10 (9), 3961-3968, 2019 | 9 | 2019 |
Synthesis and Pharmacological Evaluation of [11C]4-Methoxy-N-[2-(thiophen-2-yl)imidazo[1,2-a]pyridin-3-yl]benzamide as a Brain Penetrant PET Ligand … ET L’Estrade, HD Hansen, C Falk-Petersen, A Haugaard, N Griem-Krey, ... ACS omega 4 (5), 8846-8851, 2019 | 8 | 2019 |
Radiosynthesis and preclinical evaluation of [11C]Cimbi‐701 – Towards the imaging of cerebral 5‐HT7 receptors ET L'Estrade, V Shalgunov, FG Edgar, MG Strebl‐Bantillo, M Xiong, ... Journal of Labelled Compounds and Radiopharmaceuticals 63 (2), 46-55, 2020 | 6 | 2020 |
Accelerating PET tracer development: Establishment of a combinatorial-like, high-throughput development approach using condensation reactions and high-throughput screening EN L'Estrade, M Palner, IN Petersen, SH Keller, S Lehel, B Dall, ... EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING 43, S455-S456, 2016 | 2 | 2016 |
Optimizing the reaction conditions for the GMP production of [18F] ACI-12589, a promising candidate in the development as a PET tracer targeting α-synuclein K Bratteby, ET L’Estrade, I Dimitrakopoulos, J Molette, B Gabos, ... Nuclear Medicine and Biology 108, S87-S88, 2022 | 1 | 2022 |
Radiolabeling and in vivo evaluation of [11C]AGH-44: a potential lead structure to develop a positron emission tomography radioligand for the 5-HT7 receptor ET L’Estrade, IN Petersen, M Xiong, AS Hogendorf, A Hogendorf, ... Journal of Radioanalytical and Nuclear Chemistry 322, 847-851, 2019 | 1 | 2019 |
Fragment-based labeling using condensation reactions of six potential 5-HT7R PET tracers E Tampio L’Estrade, V Shalgunov, S Lehel, I Nymann Petersen, ... Journal of Radioanalytical and Nuclear Chemistry 326 (3), 1749-1762, 2020 | | 2020 |
F-18-Radiolabeling and in vivo evaluation of two diverse glycomimetics using PET K Bratteby, E Torkelsson, ET L'Estrade, K Peterson, V Shalgunov, ... JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS 62, S533-S534, 2019 | | 2019 |
PET radiotracer translation from rats to higher species, using an increased-throughput in vivo evaluation strategy ET L'Estrade, M Xiong, I Petersen, V Shalgunov, FG Edgar, H Hansen, ... JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS 62, S389-S390, 2019 | | 2019 |
Development and Evaluation of Potential 5-HT7 Receptor PET Tracer Candidates ET L'Estrade København: Eget forlag, 2019 | | 2019 |