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Elina T L'Estrade, Ph.D.
Elina T L'Estrade, Ph.D.
Radiochemist at Skåne University Hospital in Lund
Verified email at sund.ku.dk
Title
Cited by
Cited by
Year
The Chemogenetic Receptor Ligand Clozapine N-Oxide Induces in vivo Neuroreceptor Occupancy and Reduces Striatal Glutamate Levels
S Bærentzen, A Casado-Sainz, D Lange, V Shalgunov, IM Tejada, ...
Frontiers in Neuroscience 13, 187, 2019
412019
Improved radiosynthesis and preliminary in vivo evaluation of the 11C-labeled tetrazine [11C] AE-1 for pretargeted PET imaging
EJL Stéen, JT Jørgensen, IN Petersen, K Nørregaard, S Lehel, ...
Bioorganic & Medicinal Chemistry Letters 29 (8), 986-990, 2019
222019
In Vivo Veritas: 18F-Radiolabeled Glycomimetics Allow Insights into the Pharmacological Fate of Galectin-3 Inhibitors
K Bratteby, E Torkelsson, ET L’Estrade, K Peterson, V Shalgunov, ...
Journal of Medicinal Chemistry 63 (2), 747-755, 2019
212019
Towards selective CNS PET imaging of the 5-HT7 receptor system: Past, present and future
ET L'Estrade, M Erlandsson, FG Edgar, T Ohlsson, GM Knudsen, ...
Neuropharmacology 172, 107830, 2020
202020
Quantification accuracy of a new HRRT high throughput rat hotel using transmission-based attenuation correction: a phantom study
SH Keller, EN L'Estrade, B Dall, M Palner, M Herth
2016 IEEE Nuclear Science Symposium, Medical Imaging Conference and Room …, 2016
162016
Classics in neuroimaging: the serotonergic 2A receptor system—from discovery to modern molecular imaging
E T. L’Estrade, HD Hansen, M Erlandsson, TG Ohlsson, GM Knudsen, ...
ACS Chemical Neuroscience 9 (6), 1226-1229, 2018
142018
Blocking of efflux transporters in rats improves translational validation of brain radioligands
V Shalgunov, M Xiong, ET L’Estrade, NR Raval, IV Andersen, FG Edgar, ...
EJNMMI research 10, 1-11, 2020
122020
Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of [18F]ENL30: A Potential PET Radiotracer for the 5-HT7 Receptor
E Tampio L’Estrade, FG Edgar, M Xiong, V Shalgunov, SL Baerentzen, ...
ACS omega 4 (4), 7344-7353, 2019
112019
The α-synuclein PET tracer [18F] ACI-12589 distinguishes multiple system atrophy from other neurodegenerative diseases
R Smith, F Capotosti, M Schain, T Ohlsson, E Vokali, J Molette, ...
Nature communications 14 (1), 6750, 2023
92023
In Vitro and In Vivo Characterization of Dibenzothiophene Derivatives [125I]Iodo-ASEM and [18F]ASEM as Radiotracers of Homo- and Heteromeric α7 Nicotinic …
CK Donat, HH Hansen, HD Hansen, RC Mease, AG Horti, MG Pomper, ...
Molecules 25 (6), 1425, 2020
92020
Development and Evaluation of Two Potential 5-HT7 Receptor PET Tracers: [18F]ENL09 and [18F]ENL10
E Tampio L’Estrade, M Xiong, V Shalgunov, FG Edgar, B Volk, ...
ACS Chemical Neuroscience 10 (9), 3961-3968, 2019
92019
Synthesis and Pharmacological Evaluation of [11C]4-Methoxy-N-[2-(thiophen-2-yl)imidazo[1,2-a]pyridin-3-yl]benzamide as a Brain Penetrant PET Ligand …
ET L’Estrade, HD Hansen, C Falk-Petersen, A Haugaard, N Griem-Krey, ...
ACS omega 4 (5), 8846-8851, 2019
82019
Radiosynthesis and preclinical evaluation of [11C]Cimbi‐701 – Towards the imaging of cerebral 5‐HT7 receptors
ET L'Estrade, V Shalgunov, FG Edgar, MG Strebl‐Bantillo, M Xiong, ...
Journal of Labelled Compounds and Radiopharmaceuticals 63 (2), 46-55, 2020
62020
Accelerating PET tracer development: Establishment of a combinatorial-like, high-throughput development approach using condensation reactions and high-throughput screening
EN L'Estrade, M Palner, IN Petersen, SH Keller, S Lehel, B Dall, ...
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING 43, S455-S456, 2016
22016
Optimizing the reaction conditions for the GMP production of [18F] ACI-12589, a promising candidate in the development as a PET tracer targeting α-synuclein
K Bratteby, ET L’Estrade, I Dimitrakopoulos, J Molette, B Gabos, ...
Nuclear Medicine and Biology 108, S87-S88, 2022
12022
Radiolabeling and in vivo evaluation of [11C]AGH-44: a potential lead structure to develop a positron emission tomography radioligand for the 5-HT7 receptor
ET L’Estrade, IN Petersen, M Xiong, AS Hogendorf, A Hogendorf, ...
Journal of Radioanalytical and Nuclear Chemistry 322, 847-851, 2019
12019
Fragment-based labeling using condensation reactions of six potential 5-HT7R PET tracers
E Tampio L’Estrade, V Shalgunov, S Lehel, I Nymann Petersen, ...
Journal of Radioanalytical and Nuclear Chemistry 326 (3), 1749-1762, 2020
2020
F-18-Radiolabeling and in vivo evaluation of two diverse glycomimetics using PET
K Bratteby, E Torkelsson, ET L'Estrade, K Peterson, V Shalgunov, ...
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS 62, S533-S534, 2019
2019
PET radiotracer translation from rats to higher species, using an increased-throughput in vivo evaluation strategy
ET L'Estrade, M Xiong, I Petersen, V Shalgunov, FG Edgar, H Hansen, ...
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS 62, S389-S390, 2019
2019
Development and Evaluation of Potential 5-HT7 Receptor PET Tracer Candidates
ET L'Estrade
København: Eget forlag, 2019
2019
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