| Development and pharmacological characterization of selective blockers of 2-arachidonoyl glycerol degradation with efficacy in rodent models of multiple sclerosis and pain M Brindisi, S Maramai, S Gemma, S Brogi, A Grillo, L Di Cesare Mannelli, ... Journal of medicinal chemistry 59 (6), 2612-2632, 2016 | 79 | 2016 |
| Novel spiroindoline HDAC inhibitors: Synthesis, molecular modelling and biological studies M Brindisi, J Senger, C Cavella, A Grillo, G Chemi, S Gemma, ... European Journal of Medicinal Chemistry 157, 127-138, 2018 | 48 | 2018 |
| Structure-activity relationships, biological evaluation and structural studies of novel pyrrolonaphthoxazepines as antitumor agents M Brindisi, C Ulivieri, G Alfano, S Gemma, F de Asís Balaguer, T Khan, ... European journal of medicinal chemistry 162, 290-320, 2019 | 35 | 2019 |
| Spiroindoline-capped selective HDAC6 inhibitors: design, synthesis, structural analysis, and biological evaluation AP Saraswati, N Relitti, M Brindisi, JD Osko, G Chemi, S Federico, A Grillo, ... ACS Medicinal Chemistry Letters 11 (11), 2268-2276, 2020 | 31 | 2020 |
| Cinnamic acids derived compounds with antileishmanial activity target Leishmania amazonensis arginase ER da Silva, S Brogi, A Grillo, G Campiani, S Gemma, PC Vieira, ... Chemical Biology & Drug Design 93 (2), 139-146, 2019 | 29 | 2019 |
| Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1, 5-diarylpyrrol-3-substituted scaffold A Reale, S Brogi, A Chelini, M Paolino, A Di Capua, G Giuliani, A Cappelli, ... Bioorganic & Medicinal Chemistry 27 (19), 115045, 2019 | 24 | 2019 |
| Synthesis, Molecular Modelling and Biological Studies of 3-hydroxypyrane-4-one and 3-hydroxy-pyridine-4-one Derivatives as HIV-1 Integrase Inhibitors H Sirous, A Fassihi, S Brogi, G Campiani, F Christ, Z Debyser, S Gemma, ... Medicinal Chemistry 15 (7), 755-770, 2019 | 22 | 2019 |
| Harnessing the pyrroloquinoxaline scaffold for FAAH and MAGL interaction: definition of the structural determinants for enzyme inhibition M Brindisi, S Brogi, S Maramai, A Grillo, G Borrelli, S Butini, E Novellino, ... RSC advances 6 (69), 64651-64664, 2016 | 21 | 2016 |
| Development of novel multipotent compounds modulating endocannabinoid and dopaminergic systems A Grillo, G Chemi, S Brogi, M Brindisi, N Relitti, F Fezza, D Fazio, ... European Journal of Medicinal Chemistry 183, 111674, 2019 | 15 | 2019 |
| Structural manipulation of the conjugated phenyl moiety in 3-phenylbenzofulvene monomers: Effects on spontaneous polymerization M Paolino, G Grisci, A Reale, V Razzano, G Giuliani, A Donati, ... Polymers 10 (7), 752, 2018 | 14 | 2018 |
| Selective fatty acid amide hydrolase inhibitors as potential novel antiepileptic agents A Grillo, F Fezza, G Chemi, R Colangeli, S Brogi, D Fazio, S Federico, ... ACS Chemical Neuroscience 12 (9), 1716-1736, 2021 | 13 | 2021 |
| Development of a practical and scalable route for the preparation of the deacetoxytubuvaline (dTuv) fragment of pretubulysin and analogs M Brindisi, S Maramai, A Grillo, S Brogi, S Butini, E Novellino, G Campiani, ... Tetrahedron Letters 57 (8), 920-923, 2016 | 7 | 2016 |
| Design, synthesis, and X-ray studies of potent HIV-1 protease inhibitors with P2-carboxamide functionalities AK Ghosh, A Grillo, J Raghavaiah, S Kovela, ME Johnson, DW Kneller, ... ACS Medicinal Chemistry Letters 11 (10), 1965-1972, 2020 | 6 | 2020 |
| Small diverse antioxidant functionalities for oxidative stress disease drug discovery D Sikazwe, A Grillo, S Ramsinghani, J Davis, K McQuiston, ... Mini Reviews in Medicinal Chemistry 12 (8), 768-774, 2012 | 5 | 2012 |
| Oxalamido-substituted tricyclic inhibitors of hepatitis b virus R De Francesco, L Donnici, L Guidotti, M Iannacone, R Di Fabio, ... US Patent App. 17/611,777, 2022 | 3 | 2022 |
| Catalytic Enantioselective Diels Alder Reaction: Application in the Synthesis of Antiviral Agents A Grillo, BM Bizzarri Catalysts 12 (2), 150, 2022 | 2 | 2022 |
| Asymmetric Diels–Alder reaction of 3-(acyloxy) acryloyl oxazolidinones: optically active synthesis of a high-affinity ligand for potent HIV-1 protease inhibitors AK Ghosh, A Grillo, S Kovela, M Brindisi RSC advances 9 (71), 41755-41763, 2019 | 2 | 2019 |
| Discovery of a Novel Series of Potent SHP2 Allosteric Inhibitors A Petrocchi, A Grillo, L Ferrante, P Randazzo, A Prandi, M De Matteo, ... ACS Medicinal Chemistry Letters 14 (5), 645-651, 2023 | 1 | 2023 |
| Preparation of arylaminocarbonyl pyrrolo- fused tricyclic sulfonamides as inhibitors of hepatitis B virus R De Francesco, L Donnici, L Guidotti, M Iannacone, R Di Fabio, ... | 1 | 2019 |
| Preparation of oxalamido- substituted tricyclic inhibitors of hepatitis B virus R De Francesco, L Donnici, L Guidotti, M Iannacone, R Di Fabio, ... | 1 | 2019 |
