18F-Trifluoromethanesulfinate Enables Direct C–H 18F-Trifluoromethylation of Native Aromatic Residues in Peptides CW Kee, O Tack, F Guibbal, TC Wilson, PG Isenegger, M Imiołek, ... Journal of the American Chemical Society 142 (3), 1180-1185, 2020 | 70 | 2020 |
Manual and automated Cu-mediated radiosynthesis of the PARP inhibitor [18F]olaparib F Guibbal, PG Isenegger, TC Wilson, A Pacelli, D Mahaut, JBI Sap, ... Nature protocols 15 (4), 1525-1541, 2020 | 45 | 2020 |
Copper-Mediated Radiosynthesis of [18F]Rucaparib Z Chen, G Destro, F Guibbal, CY Chan, B Cornelissen, V Gouverneur Organic letters 23 (18), 7290-7294, 2021 | 19 | 2021 |
[18F]AZD2461, an Insight on Difference in PARP Binding Profiles for DNA Damage Response PET Imaging F Guibbal, SL Hopkins, A Pacelli, PG Isenegger, M Mosley, JB Torres, ... Molecular Imaging and Biology 22, 1226-1234, 2020 | 15 | 2020 |
Synthesis and Automated Labeling of [18F]Darapladib, a Lp-PLA2 Ligand, as Potential PET Imaging Tool of Atherosclerosis F Guibbal, V Meneyrol, I Ait-Arsa, N Diotel, J Patché, B Veeren, S Bénard, ... ACS Medicinal Chemistry Letters 10 (5), 743-748, 2019 | 15 | 2019 |
Development, synthesis, and 68Ga-Labeling of a Lipophilic complexing agent for atherosclerosis PET imaging J Yong-Sang, F Dioury, V Meneyrol, I Ait-Arsa, JP Idoumbin, F Guibbal, ... European Journal of Medicinal Chemistry 176, 129-134, 2019 | 14 | 2019 |
Imaging PARP with [18F]rucaparib in pancreatic cancer models CY Chan, Z Chen, G Destro, M Veal, D Lau, E O’Neill, G Dias, M Mosley, ... European Journal of Nuclear Medicine and Molecular Imaging 49 (11), 3668-3678, 2022 | 12 | 2022 |
Radiosynthesis of [18F]ArylSCF2H Using Aryl Boronic Acids, S-(Chlorofluoromethyl)benzenesulfonothioate and [18F]Fluoride Q Zhao, PG Isenegger, TC Wilson, JBI Sap, F Guibbal, L Lu, ... CCS Chemistry 3 (7), 1921-1028, 2021 | 9 | 2021 |
Modular construction of dynamic nucleodendrimers V Abet, R Evans, F Guibbal, S Caldarelli, R Rodriguez Angewandte Chemie International Edition 53 (19), 4862-4866, 2014 | 9 | 2014 |
A radioiodinated rucaparib analogue as an Auger electron emitter for cancer therapy G Destro, Z Chen, CY Chan, C Fraser, G Dias, M Mosley, F Guibbal, ... Nuclear Medicine and Biology 116, 108312, 2023 | 8 | 2023 |
Multi-patient dose synthesis of [18F]Flumazenil via a copper-mediated 18F-fluorination T Gendron, G Destro, NJW Straathof, JBI Sap, F Guibbal, C Vriamont, ... EJNMMI radiopharmacy and chemistry 7 (1), 5, 2022 | 7 | 2022 |
[123I] CC1: A PARP-Targeting, Auger Electron–Emitting Radiopharmaceutical for Radionuclide Therapy of Cancer CY Chan, Z Chen, F Guibbal, G Dias, G Destro, E O’Neill, M Veal, D Lau, ... Journal of Nuclear Medicine 64 (12), 1965-1971, 2023 | 4 | 2023 |
Correlation between molar activity, injection mass and uptake of the PARP targeting radiotracer [18F]olaparib in mouse models of glioma CY Chan, SL Hopkins, F Guibbal, A Pacelli, J Baguña Torres, M Mosley, ... EJNMMI research 12 (1), 67, 2022 | 4 | 2022 |
Regioselectivity of thiouracil alkylation: Application to optimization of Darapladib synthesis F Guibbal, S Bénard, J Patché, V Meneyrol, J Couprie, J Yong-Sang, ... Bioorganic & Medicinal Chemistry Letters 28 (4), 787-792, 2018 | 4 | 2018 |
Imaging PARP with 18F-rucaparib CY Chan, Z Chen, G Destro, M Veal, D Lau, E O’Neill, G Dias, M Mosley, ... Journal of Nuclear Medicine 62 (supplement 1), 1516-1516, 2021 | 1 | 2021 |
Imaging the Sirtuin 2 (SIRT2) protein-[18F] PF-SIRT, a novel positron emission tomography radioligand candidate C Read, RF Garros, F Guibbal, A Yadav, C Plisson, H Cassese, R Tucker, ... Nuclear Medicine and Biology 126, 108577, 2023 | | 2023 |
Radiolabeled darapladib and analogs thereof and their use as imaging compounds O Meilhac, E Jestin, F Guibbal, S Benard US Patent App. 18/061,715, 2023 | | 2023 |
Radiolabeled Darapladib and analogs thereof and their use as imaging compounds O Meilhac, E Jestin, F Guibbal, S Benard US Patent 11,583,596, 2023 | | 2023 |
Radiopharmaceutical for Radionuclide Therapy of Cancer CY Chan, Z Chen, F Guibbal, G Dias, G Destro, E O’Neill, M Veal, D Lau, ... | | 2023 |
Synthesis, Radiosynthesis, and In Vitro Evaluation of an Iodine-123 agent for Targeted Radionuclide Therapy of PARP-expressing Tumours G Destro, Z Chen, C Chan, G Dias, C Fraser, M Mosley, E O'Neill, ... EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING 49 (SUPPL 1 …, 2022 | | 2022 |