Examination of diazaspiro cores as piperazine bioisosteres in the olaparib framework shows reduced DNA damage and cytotoxicity SW Reilly, LN Puentes, K Wilson, CJ Hsieh, CC Weng, M Makvandi, ... Journal of medicinal chemistry 61 (12), 5367-5379, 2018 | 43 | 2018 |
A Solid‐Phase Approach to Accessing Bisthioether‐Stapled Peptides Resulting in a Potent Inhibitor of PRC2 Catalytic Activity G Zhang, F Barragan, K Wilson, N Levy, A Herskovits, M Sapozhnikov, ... Angewandte Chemie International Edition 57 (52), 17073-17078, 2018 | 20 | 2018 |
An allosteric modulator of PRC2 methyltransferase activity inhibits renal cancer cell proliferation G Gerona-Navarro, G Zhang, F Barragan, B Elie, K Wilson, A Herskovits, ... European Journal of Cancer 138, S23-S24, 2020 | | 2020 |
Solid phase synthesis of all hydrocarbon bis-thioether stapled peptides: Application to developing new inhibitors of the master transcriptional regulator EZH2 G Zhang, F Barragan, K Wilson, A Herskovits, G Gerona-Navarro ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 254, 2017 | | 2017 |