| Ambient Temperature Synthesis of High Enantiopurity N-Protected Peptidyl Ketones by Peptidyl Thiol Ester−Boronic Acid Cross-Coupling H Yang, H Li, R Wittenberg, M Egi, W Huang, LS Liebeskind Journal of the American Chemical Society 129 (5), 1132-1140, 2007 | 150 | 2007 |
| Chutes and ladders in hepatitis C nucleoside drug development SJ Coats, EC Garnier-Amblard, F Amblard, M Ehteshami, S Amiralaei, ... Antiviral research 102, 119-147, 2014 | 80 | 2014 |
| A Copper‐Catalyzed, pH‐Neutral Construction of High‐Enantiopurity Peptidyl Ketones from Peptidic S‐Acylthiosalicylamides in Air at Room Temperature LS Liebeskind, H Yang, H Li Angewandte Chemie 121 (8), 1445-1449, 2009 | 73 | 2009 |
| Synthesis of high enantiopurity N-protected α-amino ketones by thiol ester-organostannane cross-coupling using pH-neutral conditions H Li, H Yang, LS Liebeskind Organic letters 10 (19), 4375, 2008 | 73 | 2008 |
| Stereocontrolled synthesis of α-amino-α′-alkoxy ketones by a copper-catalyzed cross-coupling of peptidic thiol esters and α-alkoxyalkylstannanes H Li, A He, JR Falck, LS Liebeskind Organic letters 13 (14), 3682-3685, 2011 | 45 | 2011 |
| Computer-aided discovery and characterization of novel Ebola virus inhibitors SJ Capuzzi, W Sun, EN Muratov, C Martínez-Romero, S He, W Zhu, H Li, ... Journal of medicinal chemistry 61 (8), 3582-3594, 2018 | 38 | 2018 |
| An approach toward the alkaloid (±)-mersicarpine using a rhodium (II) carbenoid cyclization–cycloaddition cascade of an α-diazo dihydroindolinone H Li, B Cheng, N Boonnak, A Padwa Tetrahedron 67 (51), 9829-9836, 2011 | 31 | 2011 |
| Model studies directed toward the alkaloid mersicarpine utilizing a Rh (II)-catalyzed insertion/cycloaddition sequence H Li, SA Bonderoff, B Cheng, A Padwa The Journal of Organic Chemistry 79 (1), 392-400, 2014 | 25 | 2014 |
| N-Alkenyl Indoles as Useful Intermediates for Alkaloid Synthesis H Li, N Boonnak, A Padwa The Journal of Organic Chemistry 76 (22), 9488-9496, 2011 | 23 | 2011 |
| Torin 2 Derivative, NCATS-SM3710, Has Potent Multistage Antimalarial Activity through Inhibition of P. falciparum Phosphatidylinositol 4-Kinase (Pf PI4KIIIβ) K Krishnan, P Ziniel, H Li, X Huang, D Hupalo, N Gombakomba, ... ACS Pharmacology & Translational Science 3 (5), 948-964, 2020 | 19 | 2020 |
| Novel lead structures with both Plasmodium falciparum gametocytocidal and asexual blood stage activity identified from high throughput compound screening W Sun, X Huang, H Li, G Tawa, E Fisher, TQ Tanaka, P Shinn, W Huang, ... Malaria Journal 16, 1-11, 2017 | 18 | 2017 |
| Intramolecular Cycloaddition Reactions of Furo[3,4-b]indoles for Alkaloid Synthesis. CSS Albert Padwa, Yan Zou, Bo Cheng, Hao Li, Nadale Downer-Riley The Journal of Organic Chemistry 79, 3173-3184, 2014 | 14 | 2014 |
| Nucleotide substrate specificity of anti-hepatitis C virus nucleoside analogs for human mitochondrial RNA polymerase M Ehteshami, L Zhou, S Amiralaei, JR Shelton, JH Cho, H Zhang, H Li, ... Antimicrobial agents and chemotherapy 61 (8), 10.1128/aac. 00492-17, 2017 | 11 | 2017 |
| Synthesis and anti-HCV activity of β-D-2′-deoxy-2′-α-chloro-2′-β-fluoro and β-d-2′-deoxy-2′-α-bromo-2′-β-fluoro nucleosides and their phosphoramidate prodrugs R Ovadia, A Khalil, H Li, C De Schutter, S Mengshetti, S Zhou, L Bassit, ... Bioorganic & medicinal chemistry 27 (4), 664-676, 2019 | 9 | 2019 |
| Efficient Synthesis of 1,9-Substituted Benzo[h][1,6]naphthyridin-2(1H)-ones and Evaluation of their Plasmodium falciparum Gametocytocidal Activities H Li, W Sun, X Huang, X Lu, PR Patel, M Kim, MJ Orr, RM Fisher, ... ACS combinatorial science 19 (12), 748-754, 2017 | 9 | 2017 |
| Synthesis of N-vinyl substituted indoles and their acid-catalyzed behavior H Li, N Boonnak, A Padwa Tetrahedron Letters 52 (17), 2062-2064, 2011 | 8 | 2011 |
| Nucleoside analogs for treatment of the flaviviridae family of viruses and cancer SJ Coats, F Amblard, S Mengshetti, H Li, RF Schinazi US Patent 10,011,629, 2018 | 4 | 2018 |
| Synthesis and antiviral evaluation of fluorinated acyclo-nucleosides and their phosphoramidates S Mahmoud, H Li, TR McBrayer, L Bassit, SF Hammad, SJ Coats, ... Nucleosides, Nucleotides and Nucleic Acids 36 (1), 66-82, 2017 | 3 | 2017 |
| Acid‐Promoted Cascade Reaction of N‐(4‐Chloroquinolin‐3‐yl)carbamates with Amines: One‐Pot Assembly of Imidazo[4,5‐c]quinolin‐2‐ones X Lu, M Kim, MJ Orr, H Li, W Huang European journal of organic chemistry 2018 (13), 1572-1580, 2018 | 2 | 2018 |
| Compounds and method for blocking transmission of malarial parasite W Huang, H Li, W Sun, X Huang, PR Patel, H Sun, W Zheng, X Lu, ... US Patent 11,753,408, 2023 | 1 | 2023 |
