Antibacterial activity and mode of action of a sulfonamide-based class of oxaborole leucyl-tRNA-synthetase inhibitors Y Si, S Basak, Y Li, J Merino, JN Iuliano, SG Walker, PJ Tonge ACS infectious diseases 5 (7), 1231-1238, 2019 | 30 | 2019 |
Structure–kinetic relationship studies for the development of long residence time LpxC inhibitors S Basak, Y Li, S Tao, F Daryaee, J Merino, C Gu, SL Delker, JN Phan, ... Journal of medicinal chemistry 65 (17), 11854-11875, 2022 | 9 | 2022 |
Impact of target turnover on the translation of drug-target residence time to time-dependent antibacterial activity R Basu, N Wang, S Basak, F Daryaee, M Babar, EK Allen, SG Walker, ... ACS infectious diseases 7 (9), 2755-2763, 2021 | 5 | 2021 |
A Long Residence Time Enoyl-Reductase Inhibitor Explores an Extended Binding Region with Isoenzyme-Dependent Tautomer Adaptation and Differential Substrate-Binding Loop Closure S Eltschkner, J Kehrein, TA Le, S Davoodi, B Merget, S Basak, ... ACS infectious diseases 7 (4), 746-758, 2021 | 4 | 2021 |
Drug Target Residence Time and the Pharmacodynamics of Antibacterial Agents S Basak, PJ Tonge 2020 Medicinal Chemistry Reviews 55, 2020 | 2 | 2020 |
Design and Synthesis of α-Truxillic Acid-Based Fatty Acid Binding Protein Inhibitors as Anti-Nociceptive and Anti-Inflammatory Agents T Clement State University of New York at Stony Brook, 2018 | 1 | 2018 |
The Interplay between Target Turnover, Residence Time and Post Antibiotic Effect R Basu State University of New York at Stony Brook, 2021 | | 2021 |
From Ring-Opening Metathesis Polymerization (ROMP) to Alternating ROMP (AROMP): I. Blocking Cholera Toxin Internalization with ROMP Glycopolymers II. Deciphering Ring-Opening … G Youn State University of New York at Stony Brook, 2021 | | 2021 |
Development and MOA Study of Antimicrobial Agents Inhibiting Selected Protein Targets Y Si State University of New York at Stony Brook, 2018 | | 2018 |