Recent advances in the chemistry of metallated azetidines D Antermite, L Degennaro, R Luisi Organic & biomolecular chemistry 15 (1), 34-50, 2017 | 112 | 2017 |
Chemical and structural investigation of the paroxetine-human serotonin transporter complex JA Coleman, V Navratna, D Antermite, D Yang, JA Bull, E Gouaux eLife, e56427, 2020 | 62 | 2020 |
Bromomethyllithium-mediated chemoselective homologation of disulfides to dithioacetals V Pace, A Pelosi, D Antermite, O Rosati, M Curini, W Holzer Chemical Communications 52 (12), 2639-2642, 2016 | 62 | 2016 |
Regio- and Stereoselective Palladium-Catalyzed C(sp3)–H Arylation of Pyrrolidines and Piperidines with C(3) Directing Groups D Antermite, DP Affron, JA Bull Organic letters 20 (13), 3948-3952, 2018 | 54 | 2018 |
Transition Metal-Catalyzed Directed C (sp3)–H Functionalization of Saturated Heterocycles D Antermite, JA Bull Synthesis 51 (17), 3171-3204, 2019 | 48 | 2019 |
Amino-oxetanes as amide isosteres by an alternative defluorosulfonylative coupling of sulfonyl fluorides JJ Rojas, RA Croft, AJ Sterling, EL Briggs, D Antermite, DC Schmitt, ... Nature Chemistry 14 (2), 160-169, 2022 | 36 | 2022 |
Stereoselective Palladium‐Catalyzed C(sp3)−H Mono‐Arylation of Piperidines and Tetrahydropyrans with a C(4) Directing Group AS Piticari, D Antermite, JI Higham, JH Moore, MP Webster, JA Bull Advanced Synthesis & Catalysis 364 (8), 1488-1497, 2022 | 11 | 2022 |
On the Mechanism and Selectivity of Palladium-Catalyzed C(sp3)–H Arylation of Pyrrolidines and Piperidines at Unactivated C4 Positions: Discovery of an … D Antermite, AJP White, L Casarrubios, JA Bull ACS Catalysis 13, 9597-9615, 2023 | 4 | 2023 |
Late-stage synthesis of heterobifunctional molecules for PROTAC applications via ruthenium-catalysed C‒H amidation D Antermite, SD Friis, JR Johansson, OD Putra, L Ackermann, ... Nature Communications 14 (1), 8222, 2023 | | 2023 |
C(sp3)u2013H functionalization of saturated heterocycles at unactivated positions: Exploring 3D vectors for fragment growth D Antermite, J Bull, J Higham, O Davies, D Affron American Chemical Society SciMeetings 1 (2), 2020 | | 2020 |
Palladium-catalysed directed C (sp3)-H functionalisation of saturated N-heterocycles at unactivated C4 positions D Antermite Imperial College London, 2020 | | 2020 |
Pd-catalyzed C (4)-H functionalization of pyrrolidines and piperidines with C (3)-directing groups: Mechanistic insight into regio-and stereoselectivity D Antermite, J Bull ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 258, 2019 | | 2019 |
C (sp3)-H functionalization of saturated heterocycles at unactivated positions: Exploring 3D vectors for fragment growth D Antermite, D Affron, O Davis, J Bull ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 258, 2019 | | 2019 |